Novel C-Ring-Hydroxy-Substituted Controlled Deactivation Cannabinergic Analogues (Q41161167)

27 September 2017

Novel C-Ring-Hydroxy-Substituted Controlled Deactivation Cannabinergic Analogues (English)

1 reference

27 September 2017

Alexandros Makriyannis

14

object named as

Alexandros Makriyannis

1 reference

27 September 2017

Shashank Kulkarni

1

1 reference

27 September 2017

Spyros P Nikas

2

1 reference

27 September 2017

Rishi Sharma

3

1 reference

27 September 2017

Shan Jiang

4

1 reference

27 September 2017

Carol A Paronis

5

1 reference

27 September 2017

Michael Z Leonard

6

1 reference

27 September 2017

Bin Zhang

7

1 reference

27 September 2017

Chandrashekhar Honrao

8

1 reference

27 September 2017

Srikrishnan Mallipeddi

9

1 reference

27 September 2017

Jimit Girish Raghav

10

1 reference

27 September 2017

Othman Benchama

11

1 reference

27 September 2017

Torbjörn U C Järbe

12

1 reference

27 September 2017

Jack Bergman

13

1 reference

27 September 2017

language of work or name

English

0 references

publication date

1 July 2016

1 reference

Journal of Medicinal Chemistry

27 September 2017

1 reference

27 September 2017

59

1 reference

27 September 2017

14

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27 September 2017

6903-6919

1 reference

Design and synthesis of novel prostaglandin E2 ethanolamide and glycerol ester probes for the putative prostamide receptor(s)

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Medicinal chemistry of cannabinoids

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

3'-functionalized adamantyl cannabinoid receptor probes

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Probing the carboxyester side chain in controlled deactivation (-)-δ(8)-tetrahydrocannabinols

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

C-ring cannabinoid lactones: a novel cannabinergic chemotype

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

2012 Division of medicinal chemistry award address. Trekking the cannabinoid road: a personal perspective

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Enantioselective synthesis of (10S)- and (10R)-methyl-anandamides

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Controlled-deactivation cannabinergic ligands

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Diuretic effects of cannabinoid agonists in mice

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Therapeutic utility of cannabinoid receptor type 2 (CB(2)) selective agonists

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Novel adamantyl cannabinoids as CB1 receptor probes

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Cannabinoid discrimination and antagonism by CB(1) neutral and inverse agonist antagonists

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Δ(9)-Tetrahydrocannabinol acts as a partial agonist/antagonist in mice

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

The emerging role of human esterases

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Species differences in distribution and prediction of human V(ss) from preclinical data

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Role of cannabinoids in the treatment of pain and (painful) spasticity

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Novel 1',1'-chain substituted hexahydrocannabinols: 9β-hydroxy-3-(1-hexyl-cyclobut-1-yl)-hexahydrocannabinol (AM2389) a highly potent cannabinoid receptor 1 (CB1) agonist.

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Heteroadamantyl cannabinoids

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Enhancement of endocannabinoid signaling by fatty acid amide hydrolase inhibition: a neuroprotective therapeutic modality

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Cannabilactones: a novel class of CB2 selective agonists with peripheral analgesic activity

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

The diverse CB1 and CB2 receptor pharmacology of three plant cannabinoids: delta9-tetrahydrocannabinol, cannabidiol and delta9-tetrahydrocannabivarin

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

The endocannabinoid system as an emerging target of pharmacotherapy

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

The cannabinergic system as a target for anti-inflammatory therapies

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Structural requirements for cannabinoid receptor probes.

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Pharmacokinetics and pharmacodynamics of cannabinoids

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Molecular characterization of a peripheral receptor for cannabinoids

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Comparison of the pharmacology and signal transduction of the human cannabinoid CB1 and CB2 receptors

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Determination and characterization of a cannabinoid receptor in rat brain

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

A novel probe for the cannabinoid receptor

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Classical/nonclassical hybrid cannabinoids: southern aliphatic chain-functionalized C-6beta methyl, ethyl, and propyl analogues

27 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Cannabinoids. 3. Synthetic approaches to 9-ketocannabinoids. Total synthesis of nabilone

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Unsaturated side chain beta-11-hydroxyhexahydrocannabinol analogs

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5532543

Synthesis of functionalized cannabinoids

19 August 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/27367336

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

(-)-11-Hydroxy-7'-isothiocyanato-1',1'-dimethylheptyl-delta 8-THC: a novel, high-affinity irreversible probe for the cannabinoid receptor in the brain

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/27367336

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Cannabinoid receptors as therapeutic targets

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/27367336

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/ACS.JMEDCHEM.6B00717

1 reference

27 September 2017

1 reference

27 September 2017

PubMed publication ID

27367336

1 reference