Evidence for protean agonism of RX 831003 at alpha 2A-adrenoceptors by co-expression with different G alpha protein subunits (Q42521477)

1 November 2017

Evidence for protean agonism of RX 831003 at alpha 2A-adrenoceptors by co-expression with different G alpha protein subunits (English)

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1 November 2017

Pauwels PJ

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1 November 2017

Rauly I

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2

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1 November 2017

Wurch T

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1 November 2017

Colpaert FC

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4

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1 November 2017

1 May 2002

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1 November 2017

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1 November 2017

42

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1 November 2017

6

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1 November 2017

855-863

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Effector pathway-dependent relative efficacy at serotonin type 2A and 2C receptors: evidence for agonist-directed trafficking of receptor stimulus.

1 November 2017

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https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

Modulation of 5-HT1A receptor signalling by point-mutation of cysteine351 in the rat Galpha(o) protein.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

Structural instability of a constitutively active G protein-coupled receptor. Agonist-independent activation due to conformational flexibility

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

7 January 2021

Pharmacological proteus?

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https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

Agonist-receptor efficacy. II. Agonist trafficking of receptor signals

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

Inverse, protean, and ligand-selective agonism: matters of receptor conformation

7 January 2021

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https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

A three-state receptor model of agonist action

7 January 2021

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https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

Inverse agonism and the regulation of receptor number

7 January 2021

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https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

Inverse agonism: pharmacological curiosity or potential therapeutic strategy?

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

Disparate ligand-mediated Ca(2+) responses by wild-type, mutant Ser(200)Ala and Ser(204)Ala alpha(2A)-adrenoceptor: G(alpha15) fusion proteins: evidence for multiple ligand-activation binding sites

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

Heterogeneous ligand-mediated Ca(++) responses at wt and mutant alpha(2A)-adrenoceptors suggest multiple ligand activation binding sites at the alpha(2A)-adrenoceptor

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

How efficacious are 5-HT1B/D receptor ligands: an answer from GTP gamma S binding studies with stably transfected C6-glial cell lines

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

Ligand-receptor interactions as controlled by wild-type and mutant Thr(370)Lys alpha2B-adrenoceptor-Galpha15 fusion proteins

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

Modulation of ligand responses by coupling of alpha(2A)-adrenoceptors to diverse G(alpha)-proteins

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

Analysis of ligand activation of alpha 2-adrenoceptor subtypes under conditions of equal G alpha protein stoichiometry

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

Inverse agonist activity at the alpha(2A)-adrenergic receptor.

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

Characterization of G-protein alpha subunits in the Gq class: expression in murine tissues and in stromal and hematopoietic cell lines

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

G-protein activation by putative antagonists at mutant Thr373Lys alpha2A adrenergic receptors

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2801%2900201-5

10.1016/S0028-3908(01)00201-5

7 January 2021

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DOI

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1 November 2017

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