Chemistry and pharmacology of GABAB receptor ligands (Q42959792)

11 November 2017

Chemistry and pharmacology of GABAB receptor ligands (English)

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11 November 2017

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Wolfgang Froestl

1

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11 November 2017

1 January 2010

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11 November 2017

Advances in Pharmacology

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11 November 2017

58

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11 November 2017

19-62

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CGP7930: a positive allosteric modulator of the GABAB receptor.

11 November 2017

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Rapid suppression of alcohol withdrawal syndrome by baclofen.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen efficacy in reducing alcohol craving and intake: a preliminary double-blind randomized controlled study

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Suppression of alcohol delirium tremens by baclofen administration: a case report.

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen in the treatment of alcohol withdrawal syndrome: a comparative study vs diazepam

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen: a new drug for the treatment of alcohol dependence.

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Role of the GABA(B) receptor system in alcoholism and stress: focus on clinical studies and treatment perspectives

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Effectiveness and safety of baclofen for maintenance of alcohol abstinence in alcohol-dependent patients with liver cirrhosis: randomised, double-blind controlled study

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Pharmacological profiles of generalized absence seizures in lethargic, stargazer and gamma-hydroxybutyrate-treated model mice

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Double-blind randomized controlled trial of baclofen vs. clonidine in the treatment of opiates withdrawal.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

A new synthesis resolution and in vitro activities of (R)- and (S)-β-Phenyl-Gaba

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Synthesis and pharmacological evaluation of novel gamma-aminobutyric acid type B (GABAB) receptor agonists as gastroesophageal reflux inhibitors

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Reduced inhibitory action of a GABAB receptor agonist on [3H]-dopamine release from rat ventral tegmental area in vitro after chronic nicotine administration

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Distribution and properties of GABA(B) antagonist [3H]CGP 62349 binding in the rhesus monkey thalamus and basal ganglia and the influence of lesions in the reticular thalamic nucleus

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Blood-brain barrier penetration of 3-aminopropyl-n-butylphosphinic acid (CGP 36742) in rat brain by microdialysis/mass spectrometry.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Cloning and functional characterization of a gamma-hydroxybutyrate receptor identified in the human brain

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

A GABA(B) agonist reverses the behavioral sensitization to morphine in rats.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Continuous intrathecal baclofen infusion in severe spasticity after traumatic or hypoxic brain injury.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Long-term intrathecal baclofen therapy in patients with intractable spasticity

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Synthesis of the nanomolar photoaffinity GABA(B) receptor ligand CGP 71872 reveals diversity in the tissue distribution of GABA(B) receptor forms

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Gamma-hydroxybutyric acid: an endogenous neuromodulator with abuse potential?

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Different actions of gabapentin and baclofen in hippocampus from weaver mice

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Gabapentin actions on Kir3 currents and N-type Ca2+ channels via GABAB receptors in hippocampal pyramidal cells

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Molecular structure and physiological functions of GABA(B) receptors

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Attenuation of morphine withdrawal signs by the GABA(B) receptor agonist baclofen

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The heptahelical domain of GABA(B2) is activated directly by CGP7930, a positive allosteric modulator of the GABA(B) receptor

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Determination of the GABA(B) receptor agonist CGP 44532 (3-amino-2-hydroxypropylmethylphosphinic acid) in rat plasma after pre-column derivatization by micro-high-performance liquid chromatography combined with negative electrospray tandem mass spec

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Selective block of rat and human neocortex GABA(B) receptors regulating somatostatin release by a GABA(B) antagonist endowed with cognition enhancing activity

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The treatment of tetanus with intrathecal baclofen

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABAB receptor: a site of therapeutic benefit

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

(-)Baclofen decreases neurotransmitter release in the mammalian CNS by an action at a novel GABA receptor.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The GABA(B) agonist CGP 44532 decreases cocaine self-administration in rats: demonstration using a progressive ratio and a discrete trials procedure.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The GABA(B) antagonist CGP56433A attenuates the effect of baclofen on cocaine but not heroin self-administration in the rat.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Role of gamma-aminobutyric acid in antipanic drug efficacy

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Hippocampal CREB1 but not CREB2 is decreased in aged rats with spatial memory impairments

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen: a preliminary report of its pharmacological properties and therapeutic efficacy in spasticity

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The GABA(B) receptor agonist, baclofen, and the positive allosteric modulator, CGP7930, inhibit visceral pain-related responses to colorectal distension in rats.

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Epilepsy and intrathecal baclofen therapy in children with cerebral palsy

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen-mediated gastro-oesophageal acid reflux control in patients with established reflux disease

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Proconvulsive effect of the GABA(B) receptor antagonist, SCH 50911, in rats undergoing ethanol withdrawal syndrome

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Protection by the GABAB receptor antagonist, SCH 50911, of gamma-hydroxybutyric acid-induced mortality in mice

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Resuscitative effect of a gamma-aminobutyric acid B receptor antagonist on gamma-hydroxybutyric acid mortality in mice

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

In vivo effectiveness of CGP7930, a positive allosteric modulator of the GABAB receptor

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Gamma-aminobutyric acidB (GABAB)-receptor mediation of different in vivo effects of gamma-butyrolactone

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Further evidence for prejunctional GABA-B inhibition of cholinergic and peptidergic bronchoconstriction in guinea pigs: studies with new agonists and antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Novel, potent, and selective GABAC antagonists inhibit myopia development and facilitate learning and memory.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABA(C) receptor antagonists differentiate between human rho1 and rho2 receptors expressed in Xenopus oocytes.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Differential modulation by the GABAB receptor allosteric potentiator 2,6-di-tert-butyl-4-(3-hydroxy-2,2-dimethylpropyl)-phenol (CGP7930) of synaptic transmission in the rat hippocampal CA1 area

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABA(B) receptor modulators potentiate baclofen-induced depression of dopamine neuron activity in the rat ventral tegmental area

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Does gabapentin act as an agonist at native GABA(B) receptors?

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Role of GABAB receptor in alcohol dependence: Reducing effect of baclofen on alcohol intake and alcohol motivational properties in rats and amelioration of alcohol withdrawal syndrome and alcohol craving in human alcoholics

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABA(B) receptor inhibition causes locomotor stimulation in mice

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The GABA(B) receptor agonists baclofen and CGP 44532 prevent acquisition of alcohol drinking behaviour in alcohol-preferring rats

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen-induced suppression of alcohol deprivation effect in Sardinian alcohol-preferring (sP) rats exposed to different alcohol concentrations

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABA(B) receptor agonists for the treatment of drug addiction: a review of recent findings

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Unravelling the brain targets of gamma-hydroxybutyric acid

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Don't worry 'B' happy!: a role for GABA(B) receptors in anxiety and depression.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Behavioral characterization of the novel GABAB receptor-positive modulator GS39783 (N,N'-dicyclopentyl-2-methylsulfanyl-5-nitro-pyrimidine-4,6-diamine): anxiolytic-like activity without side effects associated with baclofen or benzodiazepines

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Comparative pharmacological activity of optical isomers of phenibut

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Study on brain interstitial fluid distribution and blood-brain barrier transport of baclofen in rats by microdialysis

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABA(B) receptor-mediated effects in human and rat neocortical neurones in vitro

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Intermittent intrathecal baclofen for severe tetanus

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Determination of the minimal functional ligand-binding domain of the GABAB1b receptor.

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Influence of a GABA(B) and GABA(C) receptor antagonist on sleep-waking cycle in the rat.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Antitussive effect of the GABA-agonist baclofen

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen-induced cough suppression in cervical spinal cord injury

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Treatment of chronic, refractory cough with baclofen

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

CGP 44532, a GABAB receptor agonist, is hedonically neutral and reduces cocaine-induced enhancement of reward

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen treatment for chronic posttraumatic stress disorder

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Intrathecal baclofen for spasticity

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Point mutations in the transmembrane region of GABAB2 facilitate activation by the positive modulator N,N'-dicyclopentyl-2-methylsulfanyl-5-nitro-pyrimidine-4,6-diamine (GS39783) in the absence of the GABAB1 subunit.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

A physiological role for GABAB receptors in the central nervous system.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The efficacy of intrathecal baclofen in severe tetanus

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABA(B) receptor alterations as indicators of physiological and pharmacological function

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Regulation of neurokinin-1 receptor expression by GABA(B) receptor agonists

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The role of GABA in the mediation and perception of pain

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

CGP 56999A, a GABA(B) receptor antagonist, enhances expression of brain-derived neurotrophic factor and attenuates dopamine depletion in the rat corpus striatum following a 6-hydroxydopamine lesion of the nigrostriatal pathway.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Activation of nigral dopamine neurons by the selective GABA(B)-receptor antagonist SCH 50911.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Acute interaction of baclofen in combination with alcohol in heavy social drinkers

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen antagonizes nicotine-, cocaine-, and morphine-induced dopamine release in the nucleus accumbens of rat

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen prevents drug-induced reinstatement of extinguished nicotine-seeking behaviour and nicotine place preference in rodents

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Ethanol enhances GABAB-mediated inhibitory postsynaptic transmission on rat midbrain dopaminergic neurons by facilitating GIRK currents

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Diazepam withdrawal responses measured in the social interaction test of anxiety and their reversal by baclofen

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Effects of GABA(B) receptor agents on cocaine priming, discrete contextual cue and food induced relapses.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Effects of GABA(B) receptor antagonist, agonists and allosteric positive modulator on the cocaine-induced self-administration and drug discrimination

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen for alcohol dependence: a preliminary open-label study

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The GABA B agonist baclofen reduces cigarette consumption in a preliminary double-blind placebo-controlled smoking reduction study.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Effects of imipramine or GABA(B) receptor ligands on the immobility, swimming and climbing in the forced swim test in rats following discontinuation of cocaine self-administration

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Ligands for the isolation of GABA(B) receptors [corrected] .

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Ligands for expression cloning and isolation of GABA(B) receptors

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https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

SGS742: the first GABA(B) receptor antagonist in clinical trials

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen as an adjuvant analgesic

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Comparison of L-baclofen and racemic baclofen in trigeminal neuralgia

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen in the treatment of trigeminal neuralgia: double-blind study and long-term follow-up

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen in Trigeminal Neuralgia Its Effect on the Spinal Trigeminal Nucleus: A Pilot Study

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABAB antagonists: resolution, absolute stereochemistry, and pharmacology of (R)- and (S)-phaclofen.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Conditional gene deletion reveals functional redundancy of GABAB receptors in peripheral nociceptors in vivo

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The GABA-B antagonist CGP 36742 prevent PTZ-kindling-provoked amnesia in rats.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The modulatory effects of high affinity GABA(B) receptor antagonists in an active avoidance learning paradigm in rats.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Effects of GABAB receptor antagonists on learning and memory retention in a rat model of absence epilepsy.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Effects of high-affinity GABAB receptor antagonists on active and passive avoidance responding in rodents with gamma-hydroxybutyrolactone-induced absence syndrome

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Quality of life: effect of reduced spasticity from intrathecal baclofen.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

In vivo modulation of ventral tegmental area dopamine and glutamate efflux by local GABA(B) receptors is altered after repeated amphetamine treatment

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The positive allosteric modulator GS39783 enhances GABA(B) receptor-mediated inhibition of cyclic AMP formation in rat striatum in vivo

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Receptor activation involving positive allosteric modulation, unlike full agonism, does not result in GABAB receptor desensitization

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Changes in the properties of allosteric and orthosteric GABAB receptor ligands after a continuous, desensitizing agonist pretreatment

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Involvement of gamma-hydroxybutyrate (GHB) and GABA-B receptors in the acute behavioral effects of GHB in baboons

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Chronic intragastric administration of gamma-butyrolactone produces physical dependence in baboons.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Effects of GABA-B agonist baclofen on bronchial hyperreactivity to inhaled histamine in subjects with cervical spinal cord injury

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen therapy for chronic hiccup

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Syntheses and optimization of new GS39783 analogues as positive allosteric modulators of GABA B receptors

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Therapeutic intervention in mice deficient for succinate semialdehyde dehydrogenase (gamma-hydroxybutyric aciduria)

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Effects of baclofen on cocaine self-administration: opioid- and nonopioid-dependent volunteers

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABAB receptor antagonists elevate both mRNA and protein levels of the neurotrophins nerve growth factor (NGF) and brain-derived neurotrophic factor (BDNF) but not neurotrophin-3 (NT-3) in brain and spinal cord of rats

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen enhances extinction of opiate conditioned place preference.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABAB receptor antagonist SGS742 improves spatial memory and reduces protein binding to the cAMP response element (CRE) in the hippocampus

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen for prevention of migraine.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen in cluster headache

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The use of baclofen in cluster headache

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

3H-baclofen and 3H-GABA bind to bicuculline-insensitive GABAB sites in rat brain

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Enantioselective actions of 4-amino-3-hydroxybutanoic acid and (3-amino-2-hydroxypropyl)methylphosphinic acid at recombinant GABA(C) receptors

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Novel high-affinity and selective biaromatic 4-substituted gamma-hydroxybutyric acid (GHB) analogues as GHB ligands: design, synthesis, and binding studies.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Pharmacologic rescue of lethal seizures in mice deficient in succinate semialdehyde dehydrogenase

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Cloning by functional expression of a member of the glutamate receptor family

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Attenuation of the stimulant response to ethanol is associated with enhanced ataxia for a GABA, but not a GABA, receptor agonist

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen attenuates conditioned locomotion to cues associated with cocaine administration and stabilizes extracellular glutamate levels in rat nucleus accumbens.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Evaluation of the anxiolytic-like profile of the GABAB receptor positive modulator CGP7930 in rodents

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The anticonvulsant gabapentin (neurontin) does not act through gamma-aminobutyric acid-B receptors.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Structure of the metabotropic glutamate receptor

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Hippocampal synapsin isoform levels are linked to spatial memory enhancement by SGS742.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Multi-center trial of baclofen for abstinence initiation in severe cocaine-dependent individuals

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

AMPA and GABA(B) receptor antagonists and their interaction in rats with a genetic form of absence epilepsy

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABA(B) receptors, schizophrenia and sleep dysfunction: a review of the relationship and its potential clinical and therapeutic implications

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen as adjunctive treatment for a patient with cocaine dependence and schizoaffective disorder

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Specific gamma-hydroxybutyrate-binding sites but loss of pharmacological effects of gamma-hydroxybutyrate in GABA(B)(1)-deficient mice

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Expression cloning of GABA(B) receptors uncovers similarity to metabotropic glutamate receptors

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Characterization of GABA(B) receptors involved in inhibition of motility associated with acetylcholine release in the dog small intestine: possible existence of a heterodimer of GABA(B1) and GABA(B2) subunits

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Characterisation and partial purification of the GABA(B) receptor from the rat cerebellum using the novel antagonist [3H]CGP 62349

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The (S)-enantiomer of 2-hydroxysaclofen is the active GABAB receptor antagonist in central and peripheral preparations

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

2-Hydroxy-saclofen: an improved antagonist at central and peripheral GABAB receptors

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Phaclofen: a peripheral and central baclofen antagonist.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Role of GABA transporter 3 in GABAergic synaptic transmission at striatal output neurons.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Effect of the GABA(B) agonist baclofen in patients with symptoms and duodeno-gastro-oesophageal reflux refractory to proton pump inhibitors

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Intrathecal baclofen use in adults with cerebral palsy.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Intrathecal drug administration. Present use and future trends

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Cloning, sequencing and expression of complementary DNA encoding the muscarinic acetylcholine receptor

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Structural basis of glutamate recognition by a dimeric metabotropic glutamate receptor

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Arbaclofen placarbil, a novel R-baclofen prodrug: improved absorption, distribution, metabolism, and elimination properties compared with R-baclofen.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Gabapentin is not a GABAB receptor agonist

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Phenibut (beta-phenyl-GABA): a tranquilizer and nootropic drug

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Blockade of GABA(B) receptors completely reverses age-related learning impairment.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Effects of baclofen on conditioned rewarding and discriminative stimulus effects of nicotine in rats

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Understanding and treating alcohol craving and dependence: recent pharmacological and neuroendocrinological findings

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABAB receptors as drug targets to treat gastroesophageal reflux disease

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Activation of the GABA(B) receptor inhibits transient lower esophageal sphincter relaxations in dogs

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

(R)-(3-amino-2-fluoropropyl) phosphinic acid (AZD3355), a novel GABAB receptor agonist, inhibits transient lower esophageal sphincter relaxation through a peripheral mode of action

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Effects of repeated administration of baclofen on transient lower esophageal sphincter relaxation in the dog

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Lipophilicities of baclofen ester prodrugs correlate with affinities to the ATP-dependent efflux pump P-glycoprotein: relevance for their permeation across the blood-brain barrier?

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABA(B) receptor activation in the ventral tegmental area inhibits the acquisition and expression of opiate-induced motor sensitization

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABA(B) receptors inhibit backpropagating dendritic spikes in hippocampal CA1 pyramidal cells in vivo

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Paired-pulse depression of excitatory postsynaptic current sinks in hippocampal CA1 in vivo

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABAB receptor blockade enhances theta and gamma rhythms in the hippocampus of behaving rats.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen interactions with nicotine in rats: effects on memory

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABA(B) receptor-positive modulation decreases selective molecular and behavioral effects of cocaine

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Activity-based probe for specific photoaffinity labeling gamma-aminobutyric acid B (GABAB) receptors on living cells: design, synthesis, and biological evaluation

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The GABA(B) receptor allosteric modulator CGP7930, like baclofen, reduces operant self-administration of ethanol in alcohol-preferring rats

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Control of transient lower esophageal sphincter relaxations and reflux by the GABA(B) agonist baclofen in normal subjects

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen does not alter the reinforcing, subject-rated or cardiovascular effects of intranasal cocaine in humans

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Gamma-hydroxybutyrate is a weak agonist at recombinant GABA(B) receptors.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

cDNA cloning of a serotonin 5-HT1C receptor by electrophysiological assays of mRNA-injected Xenopus oocytes

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Both GABA(B) receptor agonist and antagonists decreased brain stimulation reward in the rat.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen attenuates cue-induced reinstatement of alcohol-seeking behavior in Sardinian alcohol-preferring (sP) rats

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Reduction of alcohol's reinforcing and motivational properties by the positive allosteric modulator of the GABA(B) receptor, BHF177, in alcohol-preferring rats.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Specific reduction of alcohol's motivational properties by the positive allosteric modulator of the GABAB receptor, GS39783--comparison with the effect of the GABAB receptor direct agonist, baclofen

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Reducing effect of the positive allosteric modulator of the GABA(B) receptor, GS39,783, on alcohol self-administration in alcohol-preferring rats

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen-induced reduction of alcohol reinforcement in alcohol-preferring rats

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Altered peripheral myelination in mice lacking GABAB receptors

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABAB receptors in Schwann cells influence proliferation and myelin protein expression

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Characterization of (R,S)-5,7-di-tert-butyl-3-hydroxy-3-trifluoromethyl-3H-benzofuran-2-one as a positive allosteric modulator of GABAB receptors

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Pharmacology of absence epilepsy

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Influence of positive allosteric modulators on GABA(B) receptor coupling in rat brain: a scintillation proximity assay characterisation of G protein subtypes

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Opposite effects of a GABA(B) antagonist in two models of epileptic seizures in developing rats.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Review. Neurobiology of nicotine dependence

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Role of gamma-aminobutyric acid (GABA) and metabotropic glutamate receptors in nicotine reinforcement: potential pharmacotherapies for smoking cessation

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Is the GABA B heterodimer a good drug target?

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Sequence and expression of a metabotropic glutamate receptor

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Binding characteristics of gamma-hydroxybutyric acid as a weak but selective GABAB receptor agonist.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABA(B) receptor function and subunit expression in the rat spinal cord as indicators of stress and the antinociceptive response to antidepressants.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Amitriptyline prevents thermal hyperalgesia and modifications in rat spinal cord GABA(B) receptor expression and function in an animal model of neuropathic pain

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen in the treatment of staff‐man syndrome

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Genetic and pharmacological evidence of a role for GABA(B) receptors in the modulation of anxiety- and antidepressant-like behavior.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABAB receptor-positive modulation-induced blockade of the rewarding properties of nicotine is associated with a reduction in nucleus accumbens DeltaFosB accumulation.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Molecular cloning and characterization of the rat NMDA receptor

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen therapy for rigidity associated with Lewy body dementia.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Intrathecal baclofen for treatment of tetanus-induced spasticity

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The GABA(B) receptor antagonist CGP36742 improves learned helplessness in rats.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The GABA(B) receptor antagonist CGP36742 attenuates the baclofen- and scopolamine-induced deficit in Morris water maze task in rats

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Effect of intrathecal baclofen on bladder and sphincter function

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Gamma-aminobutyric acid type B receptors with specific heterodimer composition and postsynaptic actions in hippocampal neurons are targets of anticonvulsant gabapentin action.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

My close encounter with GABA(B) receptors

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Antidepressant-like activity of CGP 36742 and CGP 51176, selective GABAB receptor antagonists, in rodents

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABA(B) receptor antagonist CGP-36742 enhances somatostatin release in the rat hippocampus in vivo and in vitro

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Spasticity after stroke. Epidemiology and optimal treatment

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Intrathecal baclofen for long-term treatment of spasticity: a multi-centre study

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Allosteric modulation of GABA(B) receptor function in human frontal cortex.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The biological activity of d-baclofen (Lipresal®)

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

CGP 35348: a centrally active blocker of GABAB receptors

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Effect of baclofen on esophagogastric motility and gastroesophageal reflux in children with gastroesophageal reflux disease: a randomized controlled trial

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Positive regulation of GABA(B) receptors dually coupled to cyclic AMP by the allosteric agent CGP7930.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Comparative activities of the enantiomeric GABA(B) receptor agonists CGP 44532 and 44533 in central and peripheral tissues

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

CGP 36216 is a selective antagonist at GABA(B) presynaptic receptors in rat brain

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

R-(-)-beta-phenyl-GABA is a full agonist at GABAB receptors in brain slices but a partial agonist in the ileum

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Reducing effect of the positive allosteric modulators of the GABA(B) receptor, CGP7930 and GS39783, on alcohol intake in alcohol-preferring rats

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Increased GABA(B) receptor-mediated signaling reduces the susceptibility of fragile X knockout mice to audiogenic seizures

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The CGP7930 analogue 2,6-di-tert-butyl-4-(3-hydroxy-2-spiropentylpropyl)-phenol (BSPP) potentiates baclofen action at GABA(B) autoreceptors

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Gabapentin activates presynaptic GABAB heteroreceptors in rat cortical slices

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The effects of GABA(B) agonists and gabapentin on mechanical hyperalgesia in models of neuropathic and inflammatory pain in the rat.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Prolonged nicotine exposure does not alter GABA(B) receptor-mediated regulation of brain reward function.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The GABA B receptor agonists baclofen and CGP44532 decreased nicotine self-administration in the rat

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Repeated administration of the GABAB receptor agonist CGP44532 decreased nicotine self-administration, and acute administration decreased cue-induced reinstatement of nicotine-seeking in rats

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Positive modulation of GABA(B) receptors decreased nicotine self-administration and counteracted nicotine-induced enhancement of brain reward function in rats

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Intrathecal baclofen alleviates spinal cord spasticity

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Continuous intrathecal baclofen for severe spasticity

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Long-term intrathecal baclofen infusion for treatment of spasticity

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Up-regulation of GABA(B) receptors by chronic administration of the GABA(B) receptor antagonist SCH 50,911.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Chronic antidepressants and GABA "B" receptors: a GABA hypothesis of antidepressant drug action

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABAergic hypotheses of anxiety and depression: focus on GABA-B receptors

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Activation mechanism of the heterodimeric GABA(B) receptor

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Allosteric modulators of GABA(B) receptors: mechanism of action and therapeutic perspective.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Potentiation of NMDA receptor function through somatostatin release: a possible mechanism for the cognition-enhancing activity of GABA(B) receptor antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Comparison of antagonist potencies at pre- and post-synaptic GABA(B) receptors at inhibitory synapses in the CA1 region of the rat hippocampus

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Gamma-aminobutyric acid: something old, something new for bronchodilation

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Repeated administration of desipramine and a GABAB receptor antagonist, CGP 36742, discretely up-regulates GABAB receptor binding sites in rat frontal cortex

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Studies of GABA(B) receptors labelled with [(3)H]-CGP62349 in hippocampus resected from patients with temporal lobe epilepsy.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Modification of GABA(B1) and GABA(B2) receptor subunits in the somatosensory cerebral cortex and thalamus of rats with absence seizures (GAERS).

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Seizures in the developing brain result in a long-lasting decrease in GABA(B) inhibitory postsynaptic currents in the rat hippocampus

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Presynaptic metabotropic glutamate and GABAB receptors

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Gamma-hydroxybutyrate reduces mitogen-activated protein kinase phosphorylation via GABA B receptor activation in mouse frontal cortex and hippocampus

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

gamma-Hydroxybutyrate induces cyclic AMP-responsive element-binding protein phosphorylation in mouse hippocampus: an involvement of GABA(B) receptors and cAMP-dependent protein kinase activation.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Attenuation of morphine withdrawal signs by a GABAB receptor agonist in the locus coeruleus of rats

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABA(B) presynaptic receptors modulate glycine exocytosis from mouse spinal cord and hippocampus glycinergic nerve endings

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Subjective and cardiovascular effects of cocaine during treatment with amantadine and baclofen in combination

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABAB receptors within the ventral tegmental area are involved in the expression and acquisition of morphine-induced place preference in morphine-sensitized rats

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Effect of antidepressants on GABA(B) receptor function and subunit expression in rat hippocampus

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABAA and GABAB receptors modulate the K+-evoked release of sensory CGRP from the guinea pig urinary bladder

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Intrathecal baclofen for the treatment of tetanus

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

D-baclofen: Is it an antagonist at baclofen receptors?

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

D-Baclofen is an antagonist at baclofen receptors mediating antinociception in the spinal cord

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Oral baclofen in children with cerebral palsy: a double-blind cross-over pilot study

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Sequence and functional expression of the GABA A receptor shows a ligand-gated receptor super-family.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABAB receptors expressed in Xenopus oocytes by guinea pig cerebral mRNA are functionally coupled with Ca2+-dependent Cl− channels and with K+ channels, through GTP-binding proteins

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABAB receptors do not mediate the inhibitory actions of gabapentin on the spinal reflex in rats

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Intrathecal baclofen therapy in stiff-man syndrome: a double-blind, placebo-controlled trial

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The role of GABAB receptors in depression and antidepressant-related behavioural responses

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABAB receptor antagonist-mediated antidepressant-like behavior is serotonin-dependent.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The GABAB receptor-positive modulator GS39783 and the GABAB receptor agonist baclofen attenuate the reward-facilitating effects of cocaine: intracranial self-stimulation studies in the rat.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Localization of GABA(B) (R1) receptors in the rat hippocampus by immunocytochemistry and high resolution autoradiography, with specific reference to its localization in identified hippocampal interneuron subpopulations

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

High-dose oral baclofen: experience in patients with multiple sclerosis

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Effects of positive allosteric modulators of the GABAB receptor on cocaine self-administration in rats

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The GABAB receptor agonist baclofen prevents heroin-induced reinstatement of heroin-seeking behavior in rats.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Intrathecal baclofen therapy for stiff-man syndrome and progressive encephalomyelopathy with rigidity and myoclonus

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The reduction in paired-pulse inhibition in the rat hippocampus by gabapentin is independent of GABA(B) receptor receptor activation.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Cognitive enhancement by SGS742 in OF1 mice is linked to specific hippocampal protein expression.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Strain-dependent effects of SGS742 in the mouse

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Hippocampal levels of phosphorylated protein kinase A (phosphor-S96) are linked to spatial memory enhancement by SGS742.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The cognitive enhancer SGS742 does not involve major known signaling cascades in OF1 mice

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Expression of the GABABreceptor inXenopusoocytes and inhibition of the response by activation of protein kinase C

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

A Double-blind Crossover Trial of Baclofen-a New Treatment for the Unstable Bladder Syndrome

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Impaired function of GABA(B) receptors in tissues from pharmacoresistant epilepsy patients.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Effect of baclofen enantiomorphs on the spinal trigeminal nucleus and steric similarities of carbamazepine.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Synthesis and in vivo evaluation of [11C]CGP62349, a new GABAB receptor antagonist

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Dominant role of GABAB2 and Gbetagamma for GABAB receptor-mediated-ERK1/2/CREB pathway in cerebellar neurons.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

GABAB receptor activation protects neurons from apoptosis via IGF-1 receptor transactivation.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Use of baclofen in the treatment of esophageal stent-related hiccups

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

1 reference

7 January 2021

Functional mapping of GABA(B)-receptor subtypes in the thalamus

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Mechanisms of allosteric modulation at GABAB receptors by CGP7930 and GS39783: effects on affinities and efficacies of orthosteric ligands with distinct intrinsic properties.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

N,N'-Dicyclopentyl-2-methylsulfanyl-5-nitro-pyrimidine-4,6-diamine (GS39783) and structurally related compounds: novel allosteric enhancers of gamma-aminobutyric acidB receptor function.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Carrier-mediated transport of baclofen across monolayers of bovine brain endothelial cells in primary culture

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Stereoselective transport of baclofen across the blood-brain barrier in rats as determined by the unit impulse response methodology

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The effect of baclofen on gastro-oesophageal reflux, lower oesophageal sphincter function and reflux symptoms in patients with reflux disease

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Opposite effects of GABAB receptor antagonists on absences and convulsive seizures.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

The GABAB antagonist, CGP 35348, antagonizes the effects of baclofen, gamma-butyrolactone and HA 966 on rat striatal dopamine synthesis

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Effects of GABAergic modulators on food and cocaine self-administration in baboons

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Spontaneous and precipitated withdrawal after chronic intragastric administration of gamma-hydroxybutyrate (GHB) in baboons

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Attenuation of cocaine-seeking by GABA B receptor agonists baclofen and CGP44532 but not the GABA reuptake inhibitor tiagabine in baboons

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Novel cyclic gamma-hydroxybutyrate (GHB) analogs with high affinity and stereoselectivity of binding to GHB sites in rat brain.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Phenylacetic acids and the structurally related non-steroidal anti-inflammatory drug diclofenac bind to specific gamma-hydroxybutyric acid sites in rat brain.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Baclofen in treatment of the 'stiff-man' syndrome.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

From the street to the brain: neurobiology of the recreational drug gamma-hydroxybutyric acid

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Sensitivity of Xenopus oocytes to changes in extracellular pH: possible relevance to proposed expression of atypical mammalian GABAB receptors

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Suppression of epileptiform activity by GABA(B) receptors in wild type and weaver hippocampus 'in vitro'.

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Inhibition of morphine-induced amnesia in morphine-sensitized mice: involvement of dorsal hippocampal GABAergic receptors

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Control of transient lower oesophageal sphincter relaxations and reflux by the GABA(B) agonist baclofen in patients with gastro-oesophageal reflux disease

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

Inactivation of the maternal fragile X gene results in sensitization of GABAB receptor function in the offspring

1 reference

https://api.crossref.org/works/10.1016%2FS1054-3589%2810%2958002-5

7 January 2021

10.1016/S1054-3589(10)58002-5

Identifiers

DOI

1 reference

11 November 2017

1 reference

PubMed ID

20655477