Development and characterization of proteasome inhibitors (Q43022923)

12 November 2017

Development and characterization of proteasome inhibitors (English)

1 reference

12 November 2017

Kyung Bo Kim

1

1 reference

12 November 2017

Fabiana N Fonseca

series ordinal

2

1 reference

12 November 2017

Craig M Crews

series ordinal

3

1 reference

12 November 2017

language of work or name

English

0 references

publication date

1 January 2005

1 reference

12 November 2017

Methods in Enzymology

1 reference

12 November 2017

399

1 reference

12 November 2017

585-609

1 reference

Development of the proteasome inhibitor PS-341.

12 November 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Proteasome inhibitors: from research tools to drug candidates

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

The ubiquitin-proteasome pathway and proteasome inhibitors

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Ester bond-containing tea polyphenols potently inhibit proteasome activity in vitro and in vivo

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Antigen processing by the proteasome

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Lack of proteasome active site allostery as revealed by subunit-specific inhibitors

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Epoxomicin, a potent and selective proteasome inhibitor, exhibits in vivo antiinflammatory activity

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Eponemycin exerts its antitumor effect through the inhibition of proteasome function.

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Degradation of cell proteins and the generation of MHC class I-presented peptides

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Potent and selective inhibitors of the proteasome: dipeptidyl boronic acids

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Substrate binding and sequence preference of the proteasome revealed by active-site-directed affinity probes

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Coupling reagents and activation

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Covalent modification of the active site threonine of proteasomal beta subunits and the Escherichia coli homolog HslV by a new class of inhibitors

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Inhibitors of the proteasome block the degradation of most cell proteins and the generation of peptides presented on MHC class I molecules

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Displacement of housekeeping proteasome subunits by MHC-encoded LMPs: a newly discovered mechanism for modulating the multicatalytic proteinase complex

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Inhibition of the proteolytic activity of the multicatalytic proteinase complex (proteasome) by substrate-related peptidyl aldehydes.

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Inhibition of proteasome activities and subunit-specific amino-terminal threonine modification by lactacystin

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

The multicatalytic proteinase complex, a major extralysosomal proteolytic system

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Epoxomicin, a new antitumor agent of microbial origin

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Genes of the LMP/TAP cluster are associated with the human autoimmune disease vitiligo

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Isolation and structural determination of phepropeptins A, B, C, and D, new proteasome inhibitors, produced by Streptomyces sp.

16 August 2018

2 references

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

16 August 2018

https://api.crossref.org/works/10.1016%2FS0076-6879%2805%2999039-3

7 January 2021

TMC-95A, B, C, and D, novel proteasome inhibitors produced by Apiospora montagnei Sacc. TC 1093. Taxonomy, production, isolation, and biological activities.

2 references

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

16 August 2018

https://api.crossref.org/works/10.1016%2FS0076-6879%2805%2999039-3

7 January 2021

TMC-86A, B and TMC-96, new proteasome inhibitors from Streptomyces sp. TC 1084 and Saccharothrix sp. TC 1094. I. Taxonomy, fermentation, isolation, and biological activities.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Proteasome inhibition by the natural products epoxomicin and dihydroeponemycin: insights into specificity and potency.

16 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Towards subunit-specific proteasome inhibitors: synthesis and evaluation of peptide alpha',beta'-epoxyketones.

16 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Total synthesis of the potent proteasome inhibitor epoxomicin: a useful tool for understanding proteasome biology.

16 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Eponemycin analogues: syntheses and use as probes of angiogenesis.

16 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

Comparison of the effect of calpain inhibitors on two extralysosomal proteinases: the multicatalytic proteinase complex and m-calpain.

16 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2556561

1-Hydroxy-7-azabenzotriazole. An efficient peptide coupling additive

16 August 2018

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2805%2999039-3

7 January 2021

TMC-86A, B and TMC-96, new proteasome inhibitors from Streptomyces sp. TC 1084 and Saccharothrix sp. TC 1094. II. Physico-chemical properties and structure determination

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2805%2999039-3

7 January 2021

TMC-89A and B, new proteasome inhibitors from streptomyces sp. TC 1087

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2805%2999039-3

7 January 2021

N-methoxy-n-methylamides as effective acylating agents

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2805%2999039-3

7 January 2021

Eponemycin, a new antibiotic active against B16 melanoma. I. Production, isolation, structure and biological activity

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2805%2999039-3

7 January 2021

Epopromycins, Novel Cell Wall Synthesis Inhibitors of Plant Protoplast Produced by Strcptomyces sp. NK04000.

1 reference

https://api.crossref.org/works/10.1016%2FS0076-6879%2805%2999039-3

7 January 2021

Epopromycins, novel cell wall synthesis inhibitors of plant protoplast produced by Streptomyces sp. NK04000

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/16338383

12 December 2020

inferred from PubMed ID database lookup

Identifiers

DOI

10.1016/S0076-6879(05)99039-3

1 reference

12 November 2017

1 reference

12 November 2017

1 reference