Specific structural requirements for the inhibitory effect of thapsigargin on the Ca2+ ATPase SERCA. (Q44768427)

6 December 2017

Specific structural requirements for the inhibitory effect of thapsigargin on the Ca2+ ATPase SERCA. (English)

1 reference

6 December 2017

Cheng Xu

1

1 reference

6 December 2017

Hailun Ma

2

1 reference

6 December 2017

Giuseppe Inesi

3

1 reference

6 December 2017

Marwan K Al-Shawi

4

1 reference

6 December 2017

Chikashi Toyoshima

5

1 reference

6 December 2017

language of work or name

English

0 references

publication date

17 February 2004

1 reference

Journal of Biological Chemistry

6 December 2017

7

1 reference

based on heuristic

inferred from page(s)

published in

1 reference

6 December 2017

279

1 reference

6 December 2017

17

1 reference

6 December 2017

17973-17979

1 reference

Thapsigargin, a tumor promoter, discharges intracellular Ca2+ stores by specific inhibition of the endoplasmic reticulum Ca2(+)-ATPase

6 December 2017

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

Mechanism of inhibition of the calcium pump of sarcoplasmic reticulum by thapsigargin

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

Calcium - a life and death signal

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

Calcium signaling: a tale for all seasons

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

A tool coming of age: thapsigargin as an inhibitor of sarco-endoplasmic reticulum Ca(2+)-ATPases.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

Prostate-specific antigen-activated thapsigargin prodrug as targeted therapy for prostate cancer

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

Structural changes in the calcium pump accompanying the dissociation of calcium

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

Specific substitutions at amino acid 256 of the sarcoplasmic/endoplasmic reticulum Ca2+ transport ATPase mediate resistance to thapsigargin in thapsigargin-resistant hamster cells

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

MOLSCRIPT: a program to produce both detailed and schematic plots of protein structures

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

Comparison between the effects of the microsomal Ca(2+)-translocase inhibitors thapsigargin and 2,5-di-(t-butyl)-1,4-benzohydroquinone on cellular calcium fluxes

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

Biochemical, cellular, and pharmacological aspects of the multidrug transporter

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

Expression of avian Ca2+-ATPase in cultured mouse myogenic cells

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

Site-directed mutagenesis by overlap extension using the polymerase chain reaction

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

Use of chemical chaperones in the yeast Saccharomyces cerevisiae to enhance heterologous membrane protein expression: high-yield expression and purification of human P-glycoprotein

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

An improved assay for nanomole amounts of inorganic phosphate

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

The Escherichia coli FOF1 gammaM23K uncoupling mutant has a higher K0.5 for Pi. Transition state analysis of this mutant and others reveals that synthesis and hydrolysis utilize the same kinetic pathway

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

Transition State Analysis of the Coupling of Drug Transport to ATP Hydrolysis by P-glycoprotein

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

A factor preventing the major head protein of bacteriophage T4 from random aggregation

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

ADP-insensitive phosphoenzyme intermediate of sarcoplasmic reticulum Ca(2+)-ATPase has a compact conformation resistant to proteinase K, V8 protease and trypsin

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

Ca2+ -ATPase structure in the E1 and E2 conformations: mechanism, helix-helix and helix-lipid interactions

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

Drug binding in human P-glycoprotein causes conformational changes in both nucleotide-binding domains.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

Substrate-induced conformational changes in the transmembrane segments of human P-glycoprotein. Direct evidence for the substrate-induced fit mechanism for drug binding.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

Structure of the calcium pump from sarcoplasmic reticulum at 8-Å resolution

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M313263200

21 January 2018

Identifiers

DOI

10.1074/JBC.M313263200

1 reference

6 December 2017

1 reference