Synthesis and biological evaluation of [¹¹C]SB366791: a new PET-radioligand for in vivo imaging of the TRPV1 receptor. (Q48301223)

PubMed publication ID

23141549

10 February 2018

http://europepmc.org/abstract/MED/23141549

title

Synthesis and biological evaluation of [¹¹C]SB366791: a new PET-radioligand for in vivo imaging of the TRPV1 receptor (English)

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13 May 2020

7

Guy Bormans

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13 May 2020

author name string

Daisy van Veghel

1

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13 May 2020

Jan Cleynhens

2

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13 May 2020

Larry V Pearce

3

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13 May 2020

Peter M Blumberg

4

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13 May 2020

Koen Van Laere

5

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13 May 2020

Alfons Verbruggen

6

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publication date

7 November 2012

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PubMed publication ID

23141549

10 February 2018

http://europepmc.org/abstract/MED/23141549

published in

Nuclear Medicine and Biology

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13 May 2020

volume

40

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issue

1

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13 May 2020

page(s)

141-147

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Physiology and pharmacology of the vanilloid receptor

13 May 2020

cites work

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12 December 2020

TRPV1: a therapeutic target for novel analgesic drugs?

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Transient receptor potential channels as therapeutic targets

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Transient receptor potential vanilloid subfamily 1 expressed in pancreatic islet beta cells modulates insulin secretion in rats

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Vanilloid receptor-1 (VR1) is widely expressed on various epithelial and mesenchymal cell types of human skin

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Reduced anxiety, conditioned fear, and hippocampal long-term potentiation in transient receptor potential vanilloid type 1 receptor-deficient mice

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The capsaicin receptor: a heat-activated ion channel in the pain pathway

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Expression and distribution of vanilloid receptor 1 (TRPV1) in the adult rat brain

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Rapid calculation of polar molecular surface area and its application to the prediction of transport phenomena. 2. Prediction of blood-brain barrier penetration

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Measuring drug-related receptor occupancy with positron emission tomography

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12 December 2020

TRPV1 receptors in the central nervous system: potential for previously unforeseen therapeutic applications

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12 December 2020

Functional aspects and mechanisms of TRPV1 involvement in neurogenic inflammation that leads to thermal hyperalgesia

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12 December 2020

TRPV1 channels mediate long-term depression at synapses on hippocampal interneurons

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12 December 2020

Distribution of mRNA for vanilloid receptor subtype 1 (VR1), and VR1-like immunoreactivity, in the central nervous system of the rat and human

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12 December 2020

Halogenation of a capsaicin analogue leads to novel vanilloid TRPV1 receptor antagonists

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12 December 2020

Biodistribution and renal excretion of 99mTc-N,N'-bis-(Mercaptoacetamido) ethylenediamine. Effect of renal tubular transport inhibitors

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12 December 2020

Effects of the novel TRPV1 receptor antagonist SB366791 in vitro and in vivo in the rat.

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12 December 2020

Pharmacological characterization of vanilloid receptor located in the brain

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12 December 2020

AMG 9810 [(E)-3-(4-t-butylphenyl)-N-(2,3-dihydrobenzo[b][1,4] dioxin-6-yl)acrylamide], a novel vanilloid receptor 1 (TRPV1) antagonist with antihyperalgesic properties

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12 December 2020

TRP channels: a TR(I)P through a world of multifunctional cation channels

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12 December 2020

General anesthetics sensitize the capsaicin receptor transient receptor potential V1.

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12 December 2020

Functional transient receptor potential vanilloid 1 is expressed in human urothelial cells

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12 December 2020

Anti-dyskinetic effects of cannabinoids in a rat model of Parkinson's disease: role of CB(1) and TRPV1 receptors.

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12 December 2020

PET radiotracers: crossing the blood-brain barrier and surviving metabolism

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12 December 2020

Identification and characterisation of SB-366791, a potent and selective vanilloid receptor (VR1/TRPV1) antagonist.

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12 December 2020

[3H]Resiniferatoxin autoradiography in the CNS of wild-type and TRPV1 null mice defines TRPV1 (VR-1) protein distribution

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12 December 2020

N-(4-Tertiarybutylphenyl)-4-(3-chloropyridin-2-yl)tetrahydropyrazine -1(2H)-carbox-amide (BCTC), a Novel, Orally Effective Vanilloid Receptor 1 Antagonist with Analgesic Properties: I. In Vitro Characterization and Pharmacokinetic Properties

1 reference

12 December 2020

Topical capsaicin for pain management: therapeutic potential and mechanisms of action of the new high-concentration capsaicin 8% patch

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12 December 2020

Trpv1 reporter mice reveal highly restricted brain distribution and functional expression in arteriolar smooth muscle cells

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12 December 2020

Immunohistochemical localization of cannabinoid type 1 and vanilloid transient receptor potential vanilloid type 1 receptors in the mouse brain

1 reference

12 December 2020

Hot flash: TRPV channels in the brain.

1 reference

12 December 2020

Functional properties of the high-affinity TRPV1 (VR1) vanilloid receptor antagonist (4-hydroxy-5-iodo-3-methoxyphenylacetate ester) iodo-resiniferatoxin

1 reference

12 December 2020

Estimation of blood-brain barrier crossing of drugs using molecular size and shape, and H-bonding descriptors.

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12 December 2020

TRP channels: an overview

1 reference

12 December 2020

TRPing the switch on pain: an introduction to the chemistry and biology of capsaicin and TRPV1.

1 reference

12 December 2020

10.1016/J.NUCMEDBIO.2012.08.011

Identifiers

DOI

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13 May 2020

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13 May 2020

PubMed publication ID

23141549

1 reference