Gedunin- and Khivorin-Derivatives Are Small-Molecule Partial Agonists for Adhesion G Protein-Coupled Receptors GPR56/ADGRG1 and GPR114/ADGRG5. (Q52687704)

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scientific article published on 23 February 2018

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English	Gedunin- and Khivorin-Derivatives Are Small-Molecule Partial Agonists for Adhesion G Protein-Coupled Receptors GPR56/ADGRG1 and GPR114/ADGRG5.	scientific article published on 23 February 2018

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scholarly article

1 reference

Europe PubMed Central

5 May 2018

http://europepmc.org/abstract/MED/29476042

Gedunin- and Khivorin-Derivatives Are Small-Molecule Partial Agonists for Adhesion G Protein-Coupled Receptors GPR56/ADGRG1 and GPR114/ADGRG5. (English)

1 reference

Europe PubMed Central

5 May 2018

http://europepmc.org/abstract/MED/29476042

G protein-coupled receptor

1 reference

based on heuristic

inferred from title

author name string

Hannah M Stoveken

1

1 reference

Europe PubMed Central

5 May 2018

http://europepmc.org/abstract/MED/29476042

Scott D Larsen

2

1 reference

Europe PubMed Central

5 May 2018

http://europepmc.org/abstract/MED/29476042

Alan V Smrcka

3

1 reference

Europe PubMed Central

5 May 2018

http://europepmc.org/abstract/MED/29476042

Gregory G Tall

4

1 reference

Europe PubMed Central

5 May 2018

http://europepmc.org/abstract/MED/29476042

publication date

23 February 2018

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Europe PubMed Central

5 May 2018

http://europepmc.org/abstract/MED/29476042

Molecular Pharmacology

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Europe PubMed Central

5 May 2018

http://europepmc.org/abstract/MED/29476042

93

1 reference

Europe PubMed Central

5 May 2018

http://europepmc.org/abstract/MED/29476042

5

1 reference

Europe PubMed Central

5 May 2018

http://europepmc.org/abstract/MED/29476042

477-488

1 reference

Europe PubMed Central

5 May 2018

http://europepmc.org/abstract/MED/29476042

Stachel-independent modulation of GPR56/ADGRG1 signaling by synthetic ligands directed to its extracellular region

1 reference

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Mechano-dependent signaling by Latrophilin/CIRL quenches cAMP in proprioceptive neurons

1 reference

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Activation of Adhesion G Protein-coupled Receptors: AGONIST SPECIFICITY OF STACHEL SEQUENCE-DERIVED PEPTIDES.

1 reference

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Adhesion GPCRs in Tumorigenesis

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Orphan GPR110 (ADGRF1) targeted by N-docosahexaenoylethanolamine in development of neurons and cognitive function

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Dihydromunduletone Is a Small-Molecule Selective Adhesion G Protein-Coupled Receptor Antagonist

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Stalk-dependent and Stalk-independent Signaling by the Adhesion G Protein-coupled Receptors GPR56 (ADGRG1) and BAI1 (ADGRB1)

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The constitutive activity of the adhesion GPCR GPR114/ADGRG5 is mediated by its tethered agonist

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Structural Basis of Latrophilin-FLRT-UNC5 Interaction in Cell Adhesion

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The adhesion GPCR latrophilin/CIRL shapes mechanosensation.

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Adhesion G protein-coupled receptors are activated by exposure of a cryptic tethered agonist

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Structural basis of latrophilin-FLRT interaction

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International Union of Basic and Clinical Pharmacology. XCIV. Adhesion G protein-coupled receptors

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The adhesion GPCR GPR126 has distinct, domain-dependent functions in Schwann cell development mediated by interaction with laminin-211

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A tethered agonist within the ectodomain activates the adhesion G protein-coupled receptors GPR126 and GPR133

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Type IV collagen is an activating ligand for the adhesion G protein-coupled receptor GPR126

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The BAI subfamily of adhesion GPCRs: synaptic regulation and beyond

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Sticky signaling--adhesion class G protein-coupled receptors take the stage

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FLRT proteins are endogenous latrophilin ligands and regulate excitatory synapse development

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Therapeutic antibody targeting of CD97 in experimental arthritis: the role of antigen expression, shedding, and internalization on the pharmacokinetics of anti-CD97 monoclonal antibody 1B2

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Identifiers

10.1124/MOL.117.111476

1 reference

Europe PubMed Central

5 May 2018

http://europepmc.org/abstract/MED/29476042

0 references

1 reference

Europe PubMed Central

5 May 2018

http://europepmc.org/abstract/MED/29476042

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