Selective ligands for rat A3 adenosine receptors: structure-activity relationships of 1,3-dialkylxanthine 7-riboside derivatives. (Q54242505)

26 May 2018

title

Selective ligands for rat A3 adenosine receptors: structure-activity relationships of 1,3-dialkylxanthine 7-riboside derivatives. (English)

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26 May 2018

author name string

H O Kim

1

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26 May 2018

X D Ji

2

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26 May 2018

N Melman

3

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26 May 2018

M E Olah

4

1 reference

26 May 2018

G L Stiles

5

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26 May 2018

K A Jacobson

6

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26 May 2018

language of work or name

English

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publication date

1 November 1994

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26 May 2018

Journal of Medicinal Chemistry

published in

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26 May 2018

volume

37

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26 May 2018

issue

23

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26 May 2018

page(s)

4020-4030

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26 May 2018

Structure-activity relationships of 8-styrylxanthines as A2-selective adenosine antagonists

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The A3 adenosine receptor is the unique adenosine receptor which facilitates release of allergic mediators in mast cells

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[3H]CGS 21680, a selective A2 adenosine receptor agonist directly labels A2 receptors in rat brain

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Activation of phospholipase C via adenosine receptors provides synergistic signals for secretion in antigen-stimulated RBL-2H3 cells. Evidence for a novel adenosine receptor.

26 May 2018

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RDC8 codes for an adenosine A2 receptor with physiological constitutive activity

26 May 2018

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26 May 2018

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26 May 2018

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Molecular cloning and functional expression of a sheep A3 adenosine receptor with widespread tissue distribution.

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Characterization of adenosine receptors in rat brain by (?)[3H]N6-phenylisopropyladenosine

13 August 2018

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Evidence that the adenosine A3 receptor may mediate the protection afforded by preconditioning in the isolated rabbit heart

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BW-A522 blocks adenosine A3 receptor-mediated hypotensive responses in the rat

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Effect of trifluoromethyl and other substituents on activity of xanthines at adenosine receptors

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Photoisomerization of a potent and selective adenosine A2 antagonist, (E)-1,3-Dipropyl-8-(3,4-dimethoxystyryl)-7-methylxanthine

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Identifiers

DOI

10.1021/JM00049A021

1 reference

26 May 2018

PMC publication ID

5875426

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26 May 2018

PubMed publication ID

7966162

1 reference

26 May 2018