4-(4-(dimethylamino)phenyl)-1-methylpyridinium (APP+) is a fluorescent substrate for the human serotonin transporter. (Q30511824)

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21 January 2020

title

4-(4-(dimethylamino)phenyl)-1-methylpyridinium (APP+) is a fluorescent substrate for the human serotonin transporter (English)

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21 January 2020

0 references

1

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21 January 2020

Sergei Y Noskov

4

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21 January 2020

Louis J. De Felice

6

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21 January 2020

5

Sandra J Rosenthal

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21 January 2020

author name string

Igor Zdravkovic

2

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21 January 2020

Ian D Tomlinson

3

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21 January 2020

language of work or name

English

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publication date

30 January 2012

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Journal of Biological Chemistry

21 January 2020

published in

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21 January 2020

volume

287

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21 January 2020

issue

12

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21 January 2020

page(s)

8852-8863

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The high-affinity binding site for tricyclic antidepressants resides in the outer vestibule of the serotonin transporter

21 January 2020

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Tyr-95 and Ile-172 in transmembrane segments 1 and 3 of human serotonin transporters interact to establish high affinity recognition of antidepressants

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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26 November 2018

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12 December 2020

[Clinical effects of serotonin reuptake inhibitors--a review]

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Coupling of transmembrane proton gradients to platelet serotonin transport

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Identification of a single amino acid, phenylalanine 586, that is responsible for high affinity interactions of tricyclic antidepressants with the human serotonin transporter

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Identifiers

DOI

10.1074/JBC.M111.267757

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22291010%20AND%20SRC:MED&resulttype=core&format=json

21 January 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22291010%20AND%20SRC:MED&resulttype=core&format=json

21 January 2020

PubMed publication ID

22291010

1 reference