Virtual Screening as a Technique for PPAR Modulator Discovery (Q33502225)

27 July 2017

1 reference

title

Virtual Screening as a Technique for PPAR Modulator Discovery (English)

1 reference

27 July 2017

1 reference

David R Bevan

3

0 references

Josep Bassaganya-Riera

series ordinal

2

object named as

Josep Bassaganya-Riera

1 reference

27 July 2017

Stephanie N Lewis

1

1 reference

27 July 2017

2 September 2009

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27 July 2017

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27 July 2017

2010

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27 July 2017

861238

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Creative Commons Attribution 3.0 Unported

27 July 2017

start time

1 January 2010

1 reference

April 2022 Public Data File from Crossref

copyright status

copyrighted

1 reference

April 2022 Public Data File from Crossref

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21 June 2018

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21 June 2018

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21 June 2018

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A novel partial agonist of peroxisome proliferator-activated receptor-gamma (PPARgamma) recruits PPARgamma-coactivator-1alpha, prevents triglyceride accumulation, and potentiates insulin signaling in vitro

21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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A new class of peroxisome proliferator-activated receptor agonists with a novel binding epitope shows antidiabetic effects

21 June 2018

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21 June 2018

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Combining ethnopharmacology and virtual screening for lead structure discovery: COX-inhibitors as application example.

21 June 2018

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21 June 2018

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High throughput screening identifies novel inhibitors of Escherichia coli dihydrofolate reductase that are competitive with dihydrofolate

21 June 2018

1 reference

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Nuclear hormone receptor targeted virtual screening

21 June 2018

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Synthesis and biological and structural characterization of the dual-acting peroxisome proliferator-activated receptor alpha/gamma agonist ragaglitazar

21 June 2018

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Structure-based virtual screening: an overview

21 June 2018

1 reference

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Structural basis for antagonist-mediated recruitment of nuclear co-repressors by PPARalpha

21 June 2018

1 reference

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Novel tricyclic-alpha-alkyloxyphenylpropionic acids: dual PPARalpha/gamma agonists with hypolipidemic and antidiabetic activity

21 June 2018

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Virtual screening and fast automated docking methods.

21 June 2018

1 reference

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Structural determinants of ligand binding selectivity between the peroxisome proliferator-activated receptors

21 June 2018

1 reference

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Structure of the PPARalpha and -gamma ligand binding domain in complex with AZ 242; ligand selectivity and agonist activation in the PPAR family

21 June 2018

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PPARgamma : a nuclear regulator of metabolism, differentiation, and cell growth

21 June 2018

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New approaches in the treatment of type 2 diabetes

21 June 2018

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Asymmetry in the PPARgamma/RXRalpha crystal structure reveals the molecular basis of heterodimerization among nuclear receptors

21 June 2018

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Nuclear-receptor ligands and ligand-binding domains

21 June 2018

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21 June 2018

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Peroxisome proliferator-activated receptors: nuclear control of metabolism

21 June 2018

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A peroxisome proliferator-activated receptor gamma ligand inhibits adipocyte differentiation

21 June 2018

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Crystal structure of the ligand binding domain of the human nuclear receptor PPARgamma

21 June 2018

1 reference

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Ligand binding and co-activator assembly of the peroxisome proliferator-activated receptor-gamma

21 June 2018

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Differential expression of peroxisome proliferator-activated receptors (PPARs): tissue distribution of PPAR-alpha, -beta, and -gamma in the adult rat

21 June 2018

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A dynamic mechanism of nuclear receptor activation and its perturbation in a human disease.

21 June 2018

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Design and synthesis of alpha-aryloxyphenylacetic acid derivatives: a novel class of PPARalpha/gamma dual agonists with potent antihyperglycemic and lipid modulating activity

21 January 2018

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Indol-1-yl acetic acids as peroxisome proliferator-activated receptor agonists: design, synthesis, structural biology, and molecular docking studies

21 January 2018

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Design and synthesis of novel N-sulfonyl-2-indole carboxamides as potent PPAR-gamma binding agents with potential application to the treatment of osteoporosis

21 January 2018

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Structural basis for the structure-activity relationships of peroxisome proliferator-activated receptor agonists

21 January 2018

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Protein flexibility in ligand docking and virtual screening to protein kinases.

21 January 2018

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Virtual screening—an overview

21 January 2018

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Binding analyses between Human PPARgamma-LBD and ligands

21 January 2018

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Sulfonylureas and Glinides Exhibit Peroxisome Proliferator-Activated Receptor Activity: A Combined Virtual Screening and Biological Assay Approach

21 January 2018

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The continuing epidemics of obesity and diabetes in the United States

21 January 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2738858

Computational Screening of Phthalate Monoesters for Binding to PPARγ

31 October 2018

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Structure-based design of indole propionic acids as novel PPARalpha/gamma co-agonists

21 January 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/19746174

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1155/2010/861238

1 reference

27 July 2017

1 reference

27 July 2017

1 reference

PubMed ID

19746174