A type 1 cholecystokinin receptor mutant that mimics the dysfunction observed for wild type receptor in a high cholesterol environment (Q34073933)

30 July 2017

title

A type 1 cholecystokinin receptor mutant that mimics the dysfunction observed for wild type receptor in a high cholesterol environment (English)

1 reference

30 July 2017

1 reference

Aditya J Desai

1

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30 July 2017

Kaleeckal G Harikumar

series ordinal

2

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30 July 2017

Laurence J Miller

series ordinal

3

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30 July 2017

language of work or name

English

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publication date

13 May 2014

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Journal of Biological Chemistry

30 July 2017

published in

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30 July 2017

volume

289

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30 July 2017

issue

26

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30 July 2017

page(s)

18314-18326

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Cholecystokinin and pancreatic cancer: the chicken or the egg?

30 July 2017

cites work

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28 July 2018

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Membrane cholesterol affects stimulus-activity coupling in type 1, but not type 2, CCK receptors: use of cell lines with elevated cholesterol.

28 July 2018

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Sensitivity of cholecystokinin receptors to membrane cholesterol content

28 July 2018

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28 July 2018

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Differential sensitivity of types 1 and 2 cholecystokinin receptors to membrane cholesterol

28 July 2018

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28 July 2018

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Synthesis and in vitro characterization of radioiodinatable benzodiazepines selective for type 1 and type 2 cholecystokinin receptors

28 July 2018

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Benzodiazepine ligands can act as allosteric modulators of the Type 1 cholecystokinin receptor

28 July 2018

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A Specific Cholesterol Binding Site Is Established by the 2.8 Å Structure of the Human β2-Adrenergic Receptor

28 July 2018

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Mutational analysis of the conserved Asp2.50 and ERY motif reveals signaling bias of the urotensin II receptor

28 July 2018

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28 July 2018

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28 July 2018

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Novel benzodiazepine photoaffinity probe stereoselectively labels a site deep within the membrane-spanning domain of the cholecystokinin receptor

28 July 2018

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Charged residues of the conserved DRY triplet of the vasopressin V1a receptor provide molecular determinants for cell surface delivery and internalization

28 July 2018

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28 July 2018

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Differential effects of modification of membrane cholesterol and sphingolipids on the conformation, function, and trafficking of the G protein-coupled cholecystokinin receptor

28 July 2018

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Distinct molecular mechanisms for agonist peptide binding to types A and B cholecystokinin receptors demonstrated using fluorescence spectroscopy

28 July 2018

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A RAPID METHOD OF TOTAL LIPID EXTRACTION AND PURIFICATION

28 July 2018

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The Role of a Conserved Region of the Second Intracellular Loop in AT1 Angiotensin Receptor Activation and Signaling

28 July 2018

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Molecular basis of agonist binding to the type A cholecystokinin receptor

28 July 2018

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28 July 2018

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28 July 2018

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28 July 2018

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28 July 2018

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An arginine residue conserved in most G protein-coupled receptors is essential for the function of the m1 muscarinic receptor.

28 July 2018

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28 July 2018

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28 July 2018

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28 July 2018

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Regulation of cytosolic acetoacetyl coenzyme A thiolase, 3-hydroxy-3-methylglutaryl coenzyme A synthase, 3-hydroxy-3-methylglutaryl coenzyme A reductase, and mevalonate kinase by low density lipoprotein and by 25-hydroxycholesterol in Chinese hamste

28 July 2018

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28 July 2018

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Use of N,O-bis-Fmoc-d-Tyr-ONSu for introduction of an oxidative iodination site into cholecystokinin family peptides

28 July 2018

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Gallbladder contraction in patients with pigment and cholesterol stones.

28 July 2018

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Characterization of two novel cholecystokinin tetrapeptide (30-33) analogues, A-71623 and A-70874, that exhibit high potency and selectivity for cholecystokinin-A receptors.

28 July 2018

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Analysis and refinement of criteria for predicting the structure and relative orientations of transmembranal helical domains

28 July 2018

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Immunochemical studies on cholecystokinin. II. Distribution and molecular heterogeneity in the central nervous system and small intestine of man and hog.

28 July 2018

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2-Substituted piperazine-derived imidazole carboxamides as potent and selective CCK1R agonists for the treatment of obesity

28 July 2018

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https://api.crossref.org/works/10.1074%2FJBC.M114.570200

1,4-Benzodiazepine peripheral cholecystokinin (CCK-A) receptor agonists

21 January 2018

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https://api.crossref.org/works/10.1074%2FJBC.M114.570200

Stimulation of cholecystokinin-A receptors with GI181771X does not cause weight loss in overweight or obese patients

21 January 2018

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https://api.crossref.org/works/10.1074%2FJBC.M114.570200

Crystal structure of rhodopsin: A G protein-coupled receptor

21 January 2018

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Role of the conserved DRY motif on G protein activation of rat angiotensin II receptor type 1A

21 January 2018

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Heterodimerization of Type A and B Cholecystokinin Receptors Enhance Signaling and Promote Cell Growth

21 January 2018

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https://api.crossref.org/works/10.1074%2FJBC.M114.570200

Differential docking of high-affinity peptide ligands to type A and B cholecystokinin receptors demonstrated by photoaffinity labeling

21 January 2018

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Fluorescent indicators distributed throughout the pharmacophore of cholecystokinin provide insights into distinct modes of binding and activation of type A and B cholecystokinin receptors.

21 January 2018

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Loxiglumide, a CCK-A receptor antagonist, stimulates calorie intake and hunger feelings in humans

21 January 2018

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Excess membrane cholesterol alters human gallbladder muscle contractility and membrane fluidity

28 October 2018

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12 December 2020

The role of the cholecystokinin-B/gastrin receptor transmembrane domains in determining affinity for subtype-selective ligands

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12 December 2020

Discovery of imidazole carboxamides as potent and selective CCK1R agonists

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12 December 2020

Defect of receptor-G protein coupling in human gallbladder with cholesterol stones

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12 December 2020

Membrane cholesterol modulates galanin-GalR2 interaction

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12 December 2020

Fluorometric method for the enzymatic determination of cholesterol

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12 December 2020

Both low- and high-affinity CCK receptor states mediate trophic effects on rat pancreatic acinar cells

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12 December 2020

CCK receptor dysfunction in muscle membranes from human gallbladders with cholesterol stones

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12 December 2020

Membrane cholesterol alters gallbladder muscle contractility in prairie dogs

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12 December 2020

Peripheral-type benzodiazepine receptor function in cholesterol transport. Identification of a putative cholesterol recognition/interaction amino acid sequence and consensus pattern

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12 December 2020

Direct G protein activation reverses impaired CCK signaling in human gallbladders with cholesterol stones

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12 December 2020

Identifiers

DOI

10.1074/JBC.M114.570200

1 reference

30 July 2017

1 reference

30 July 2017

1 reference