OGA inhibition by GlcNAc-selenazoline (Q34411395)

2 August 2017

title

OGA inhibition by GlcNAc-selenazoline (English)

1 reference

2 August 2017

7

Paul R. Rablen

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20822912

8 July 2024

author name string

Eun Ju Kim

1

1 reference

2 August 2017

Etzer Darout

3

1 reference

2 August 2017

Mohannad Abdo

4

1 reference

2 August 2017

Brian Rempel

5

1 reference

2 August 2017

Spencer Knapp

9

1 reference

2 August 2017

Dona C. Love

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20822912

8 July 2024

Stephen G. Withers

6

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20822912

8 July 2024

John A. Hanover

8

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20822912

8 July 2024

language of work or name

English

0 references

publication date

11 August 2010

1 reference

full work available at URL

2 August 2017

https://works.swarthmore.edu/cgi/viewcontent.cgi?article=1089&context=fac-chemistry

file format

Portable Document Format

online access status

open access

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20822912

https://europepmc.org/articles/PMC4210863

8 July 2024

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20822912

https://europepmc.org/articles/PMC4210863?pdf=render

8 July 2024

file format

Portable Document Format

online access status

open access

content deliverer

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20822912

https://doi.org/10.1016/j.bmc.2010.08.010

8 July 2024

online access status

open access

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20822912

https://api.elsevier.com/content/article/PII:S0968089610007479?httpAccept=text/xml

8 July 2024

1 reference

Crossref

https://api.crossref.org/works/10.1016/J.BMC.2010.08.010

https://api.elsevier.com/content/article/PII:S0968089610007479?httpAccept=text/plain

8 July 2024

1 reference

Crossref

https://api.crossref.org/works/10.1016/J.BMC.2010.08.010

Bioorganic & Medicinal Chemistry

8 July 2024

published in

1 reference

2 August 2017

volume

18

1 reference

2 August 2017

issue

19

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2 August 2017

page(s)

7058-7064

1 reference

Enhanced Nrf2-dependent induction of glutathione in mouse embryonic fibroblasts by isoselenocyanate analog of sulforaphane

2 August 2017

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Elevation of Global O-GlcNAc Levels in 3T3-L1 Adipocytes by Selective Inhibition of O-GlcNAcase Does Not Induce Insulin Resistance

6 July 2018

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O-GlcNAc regulates FoxO activation in response to glucose

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O-GlcNAc modification of FoxO1 increases its transcriptional activity: a role in the glucotoxicity phenomenon?

6 July 2018

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6 July 2018

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O-glycosylation of FoxO1 increases its transcriptional activity towards the glucose 6-phosphatase gene

6 July 2018

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Structure of N-acetyl-beta-D-glucosaminidase (GcnA) from the endocarditis pathogen Streptococcus gordonii and its complex with the mechanism-based inhibitor NAG-thiazoline

6 July 2018

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Analysis of PUGNAc and NAG-thiazoline as transition state analogues for human O-GlcNAcase: mechanistic and structural insights into inhibitor selectivity and transition state poise

6 July 2018

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Enzymatic characterization of O-GlcNAcase isoforms using a fluorogenic GlcNAc substrate

6 July 2018

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Structure and mechanism of a bacterial beta-glucosaminidase having O-GlcNAcase activity

6 July 2018

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Structural insights into the mechanism and inhibition of eukaryotic O-GlcNAc hydrolysis

6 July 2018

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Location and characterization of the O-GlcNAcase active site

6 July 2018

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The hexosamine signaling pathway: deciphering the "O-GlcNAc code"

6 July 2018

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O-GlcNAc modification on IRS-1 and Akt2 by PUGNAc inhibits their phosphorylation and induces insulin resistance in rat primary adipocytes

6 July 2018

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Isosteric replacement of sulfur with other chalcogens in peptides and proteins

6 July 2018

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O-GlcNAc modification is an endogenous inhibitor of the proteasome

6 July 2018

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Recruitment of O-GlcNAc transferase to promoters by corepressor mSin3A: coupling protein O-GlcNAcylation to transcriptional repression

6 July 2018

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Altered glycan-dependent signaling induces insulin resistance and hyperleptinemia

6 July 2018

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Regulated transport of the glucose transporter GLUT4

6 July 2018

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6 July 2018

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Hyperglycemia inhibits endothelial nitric oxide synthase activity by posttranslational modification at the Akt site

6 July 2018

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Glycan-dependent signaling: O-linked N-acetylglucosamine

6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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27 October 2018

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27 October 2018

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27 October 2018

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27 October 2018

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Comparison of biochemical parameters of benzamide riboside, a new inhibitor of IMP dehydrogenase, with tiazofurin and selenazofurin.

27 October 2018

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27 October 2018

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12 December 2020

Synthesis, structure, and antiproliferative activity of selenophenfurin, an inosine 5'-monophosphate dehydrogenase inhibitor analogue of selenazofurin

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12 December 2020

New reactions of selenocarboxylates

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12 December 2020

An O-GlcNAcase-specific inhibitor and substrate engineered by the extension of the N-acetyl moiety

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Tautomeric modification of GlcNAc-thiazoline

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Organo-phosphorus–selenium heterocycles

21

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Crossref

https://api.crossref.org/works/10.1016/J.BMC.2010.08.010

8 July 2024

Identifiers

1 reference

2 August 2017

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2 August 2017

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