Direct measurement of thermal stability of expressed CCR5 and stabilization by small molecule ligands. (Q34571010)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21155586%20AND%20SRC:MED&resulttype=core&format=json

18 January 2020

title

Direct measurement of thermal stability of expressed CCR5 and stabilization by small molecule ligands (English)

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18 January 2020

4

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18 January 2020

Thomas Huber

5

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18 January 2020

author name string

Adam M Knepp

1

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18 January 2020

Amy Grunbeck

2

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18 January 2020

Sourabh Banerjee

3

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18 January 2020

language of work or name

English

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publication date

30 December 2010

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18 January 2020

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18 January 2020

volume

50

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18 January 2020

issue

4

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18 January 2020

page(s)

502-511

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NMR analyses of the interaction between CCR5 and its ligand using functional reconstitution of CCR5 in lipid bilayers.

18 January 2020

cites work

1 reference

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7 July 2018

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Detergent screening of a G-protein-coupled receptor using serial and array biosensor technologies

7 July 2018

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Chemokine receptor antagonists: overcoming developmental hurdles

7 July 2018

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A homogeneous resonance energy transfer-based assay to monitor MutS/DNA interactions

7 July 2018

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Structural diversity of G protein-coupled receptors and significance for drug discovery

7 July 2018

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Microscale fluorescent thermal stability assay for membrane proteins

7 July 2018

1 reference

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Conformational thermostabilization of the beta1-adrenergic receptor in a detergent-resistant form

7 July 2018

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Molecular interactions of CCR5 with major classes of small-molecule anti-HIV CCR5 antagonists

7 July 2018

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Targeting chemokine receptors in HIV: a status report

7 July 2018

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Monomeric G protein-coupled receptor rhodopsin in solution activates its G protein transducin at the diffusion limit

7 July 2018

1 reference

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A monomeric G protein-coupled receptor isolated in a high-density lipoprotein particle efficiently activates its G protein

7 July 2018

1 reference

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Production and characterization of monoclonal antibodies sensitive to conformation in the 5HT2c serotonin receptor.

7 July 2018

1 reference

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Physiological roles of G protein-coupled receptor kinases and arrestins

7 July 2018

1 reference

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Chemokine: receptor structure, interactions, and antagonism

7 July 2018

1 reference

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Interaction of small molecule inhibitors of HIV-1 entry with CCR5.

7 July 2018

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HIV and the chemokine system: 10 years later

7 July 2018

1 reference

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Discovery and characterization of vicriviroc (SCH 417690), a CCR5 antagonist with potent activity against human immunodeficiency virus type 1

7 July 2018

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Maraviroc (UK-427,857), a potent, orally bioavailable, and selective small-molecule inhibitor of chemokine receptor CCR5 with broad-spectrum anti-human immunodeficiency virus type 1 activity

7 July 2018

1 reference

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Identification of a linear peptide recognized by monoclonal antibody 2D7 capable of generating CCR5-specific antibodies with human immunodeficiency virus-neutralizing activity

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3038255

Functional characterization of rhodopsin monomers and dimers in detergents

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3038255

Use of a small molecule CCR5 inhibitor in macaques to treat simian immunodeficiency virus infection or prevent simian-human immunodeficiency virus infection.

7 July 2018

1 reference

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Retinal counterion switch in the photoactivation of the G protein-coupled receptor rhodopsin

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3038255

Analysis of the mechanism by which the small-molecule CCR5 antagonists SCH-351125 and SCH-350581 inhibit human immunodeficiency virus type 1 entry.

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3038255

HIV-1 escape from a small molecule, CCR5-specific entry inhibitor does not involve CXCR4 use

7 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3038255

Development of a binding assay for p53/HDM2 by using homogeneous time-resolved fluorescence.

7 July 2018

1 reference

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Enhanced expression, native purification, and characterization of CCR5, a principal HIV-1 coreceptor

7 July 2018

1 reference

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Use of a phosphotyrosine-antibody pair as a general detection method in homogeneous time-resolved fluorescence: application to human immunodeficiency viral protease

7 July 2018

1 reference

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Epitope mapping of CCR5 reveals multiple conformational states and distinct but overlapping structures involved in chemokine and coreceptor function

7 July 2018

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Interaction of chemokine receptor CCR5 with its ligands: multiple domains for HIV-1 gp120 binding and a single domain for chemokine binding

7 July 2018

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Inhibition of human immunodeficiency virus fusion by a monoclonal antibody to a coreceptor (CXCR4) is both cell type and virus strain dependent.

7 July 2018

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Rare earth cryptates and homogeneous fluoroimmunoassays with human sera

7 July 2018

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Probing molecular interactions with homogeneous techniques based on rare earth cryptates and fluorescence energy transfer.

7 July 2018

1 reference

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Expression of a synthetic bovine rhodopsin gene in monkey kidney cells

7 July 2018

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Toward efficient drug screening by homogeneous assays based on the development of new fluorescent vasopressin and oxytocin receptor ligands.

7 July 2018

1 reference

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Probing the existence of G protein-coupled receptor dimers by positive and negative ligand-dependent cooperative binding.

27 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3038255

Cell surface detection of membrane protein interaction with homogeneous time-resolved fluorescence resonance energy transfer technology

27 October 2018

1 reference

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Allophycocyanin 1 as a near-infrared fluorescent tracer: isolation, characterization, chemical modification, and use in a homogeneous fluorescence resonance energy transfer system

27 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3038255

Tyrosine sulfation of the amino terminus of CCR5 facilitates HIV-1 entry

27 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3038255

Europium(III) trisbipyridine cryptate label for time-resolved fluorescence detection of polymerase chain reaction products fixed on a solid support.

27 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3038255

Solubilization, stabilization, and purification of chemokine receptors using biosensor technology

27 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21155586

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Analyzing ligand and small molecule binding activity of solubilized GPCRs using biosensor technology

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21155586

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Rapid Incorporation of Functional Rhodopsin into Nanoscale Apolipoprotein Bound Bilayer (NABB) Particles

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21155586

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/BI101059W

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21155586%20AND%20SRC:MED&resulttype=core&format=json

18 January 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21155586%20AND%20SRC:MED&resulttype=core&format=json

18 January 2020

PubMed publication ID

21155586

1 reference