Exploring distal regions of the A3 adenosine receptor binding site: sterically constrained N6-(2-phenylethyl)adenosine derivatives as potent ligands. (Q36342342)

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English	Exploring distal regions of the A3 adenosine receptor binding site: sterically constrained N6-(2-phenylethyl)adenosine derivatives as potent ligands.	scientific article

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27 December 2019

Exploring distal regions of the A3 adenosine receptor binding site: sterically constrained N6-(2-phenylethyl)adenosine derivatives as potent ligands (English)

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Kenneth A. Jacobson

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Zhan-Guo Gao

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Ariel S Gross

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Susanna Tchilibon

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Susanna Tchilibon

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Neli Melman

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Soo-Kyung Kim

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Brian A Harris

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Joshua B Blaustein

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Heng T Duong

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1 May 2004

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Bioorganic & Medicinal Chemistry

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2021-2034

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27 December 2019

Structural determinants of efficacy at A3 adenosine receptors: modification of the ribose moiety.

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N6-Substituted adenosine derivatives: selectivity, efficacy, and species differences at A3 adenosine receptors

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Identification of Essential Residues Involved in the Allosteric Modulation of the Human A3Adenosine Receptor

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10.1016/J.BMC.2004.02.037

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27 December 2019

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27 December 2019

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