Extending foldamer design beyond α-helix mimicry: α/β-peptide inhibitors of vascular endothelial growth factor signaling. (Q41916714)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22548447%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

title

Extending foldamer design beyond α-helix mimicry: α/β-peptide inhibitors of vascular endothelial growth factor signaling (English)

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30 January 2020

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4

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30 January 2020

author name string

Holly S Haase

1

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30 January 2020

Kimberly J Peterson-Kaufman

2

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30 January 2020

Sheeny K Lan Levengood

3

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30 January 2020

William L Murphy

5

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30 January 2020

Samuel H Gellman

6

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30 January 2020

language of work or name

English

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publication date

1 May 2012

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Journal of the American Chemical Society

30 January 2020

published in

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30 January 2020

volume

134

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30 January 2020

issue

18

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30 January 2020

page(s)

7652-7655

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Peptide and peptoid foldamers in medicinal chemistry

30 January 2020

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5 June 2018

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Interplay among side chain sequence, backbone composition, and residue rigidification in polypeptide folding and assembly

5 June 2018

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5 June 2018

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5 June 2018

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5 June 2018

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5 June 2018

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5 June 2018

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5 June 2018

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5 June 2018

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5 June 2018

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5 June 2018

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5 June 2018

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5 June 2018

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5 June 2018

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5 June 2018

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5 June 2018

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5 June 2018

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5 June 2018

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5 June 2018

1 reference

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Melanoma peptide MART-1(27-35) analogues with enhanced binding capacity to the human class I histocompatibility molecule HLA-A2 by introduction of a beta-amino acid residue: implications for recognition by tumor-infiltrating lymphocytes.

5 June 2018

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Vascular-specific growth factors and blood vessel formation

5 June 2018

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Novel peptides selected to bind vascular endothelial growth factor target the receptor-binding site

5 June 2018

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Crystal structure at 1.7 A resolution of VEGF in complex with domain 2 of the Flt-1 receptor

5 June 2018

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Vascular endothelial growth factor: crystal structure and functional mapping of the kinase domain receptor binding site

5 June 2018

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High-resolution epitope mapping of hGH-receptor interactions by alanine-scanning mutagenesis

5 June 2018

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5 June 2018

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N-alkylated oligoamide alpha-helical proteomimetics

18 August 2018

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Using a beta-hairpin to mimic an alpha-helix: cyclic peptidomimetic inhibitors of the p53-HDM2 protein-protein interaction

18 August 2018

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Design of a protein surface antagonist based on alpha-helix mimicry: inhibition of gp41 assembly and viral fusion

18 August 2018

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Requirements for binding and signaling of the kinase domain receptor for vascular endothelial growth factor

18 August 2018

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18 August 2018

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12 December 2020

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12 December 2020

Advances in the assessment and control of the effector functions of therapeutic antibodies

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12 December 2020

Expression of biologically active isoforms of the tumor angiogenesis factor VEGF in Escherichia coli

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12 December 2020

Probing the structural requirements of peptoids that inhibit HDM2-p53 interactions

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12 December 2020

Mapping of the Sites Involved in Ligand Association and Dissociation at the Extracellular Domain of the Kinase Insert Domain-containing Receptor for Vascular Endothelial Growth Factor

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Identifiers

DOI

10.1021/JA302469A

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22548447%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22548447%20AND%20SRC:MED&resulttype=core&format=json

30 January 2020

PubMed publication ID

22548447

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22548447%20AND%20SRC:MED&resulttype=core&format=json