Phenotypic screening and fragment-based approaches to the discovery of small-molecule bromodomain ligands. (Q38182138)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24467243%20AND%20SRC:MED&resulttype=core&format=json

6 March 2020

title

Phenotypic screening and fragment-based approaches to the discovery of small-molecule bromodomain ligands (English)

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6 March 2020

4

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6 March 2020

author name string

Laura E Jennings

series ordinal

1

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6 March 2020

Angelina R Measures

series ordinal

2

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6 March 2020

Brian G Wilson

series ordinal

3

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6 March 2020

publication date

1 February 2014

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Future Medicinal Chemistry

6 March 2020

published in

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6 March 2020

volume

6

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6 March 2020

issue

2

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6 March 2020

page(s)

179-204

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Selective small molecules blocking HIV-1 Tat and coactivator PCAF association

6 March 2020

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Structural basis of lysine-acetylated HIV-1 Tat recognition by PCAF bromodomain

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21 January 2018

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21 January 2018

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Identifiers

DOI

10.4155/FMC.13.197

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24467243%20AND%20SRC:MED&resulttype=core&format=json

6 March 2020

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