Synthesis of sansalvamide A peptidomimetics: triazole, oxazole, thiazole, and pseudoproline containing compounds. (Q40666063)

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21 January 2020

title

Synthesis of sansalvamide A peptidomimetics: triazole, oxazole, thiazole, and pseudoproline containing compounds (English)

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21 January 2020

6

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Katrina A. Jolliffe

9

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author name string

Melinda R Davis

1

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21 January 2020

Erinprit K Singh

2

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21 January 2020

Hendra Wahyudi

3

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21 January 2020

Leslie D Alexander

4

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21 January 2020

Joseph B Kunicki

5

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21 January 2020

Kelly A Fairweather

7

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Andrew M Giltrap

8

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Shelli R McAlpine

10

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publication date

1 January 2012

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21 January 2020

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21 January 2020

volume

68

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21 January 2020

issue

4

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page(s)

1029-1051

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Design and synthesis of Hsp90 inhibitors: exploring the SAR of Sansalvamide A derivatives

21 January 2020

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Comprehensive study of sansalvamide A derivatives and their structure-activity relationships against drug-resistant colon cancer cell lines.

22 September 2017

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Identification of Sansalvamide a analog potent against pancreatic cancer cell lines

22 September 2017

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The platelet-derived growth factor receptor alpha is destabilized by geldanamycins in cancer cells.

22 September 2017

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Hsp90 inhibitors cause G2/M arrest associated with the reduction of Cdc25C and Cdc2 in lung cancer cell lines

22 September 2017

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Involvement of calcium in the differential induction of heat shock protein 70 by heat shock protein 90 inhibitors, geldanamycin and radicicol, in human non-small cell lung cancer H460 cells

22 September 2017

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In vivo antitumor efficacy of 17-DMAG (17-dimethylaminoethylamino-17-demethoxygeldanamycin hydrochloride), a water-soluble geldanamycin derivative

22 September 2017

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Clinical Development of 17-Allylamino, 17-Demethoxygeldanamycin

22 September 2017

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Crystal structure and molecular modeling of 17-DMAG in complex with human Hsp90

22 September 2017

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Hsp90 inhibitors as novel cancer chemotherapeutic agents

22 September 2017

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Click Chemistry: Diverse Chemical Function from a Few Good Reactions

22 September 2017

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22 September 2017

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22 September 2017

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22 September 2017

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25 September 2017

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Mechanistic studies of Sansalvamide A-amide: an allosteric modulator of Hsp90.

15 June 2018

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Synthesis of second-generation sansalvamide A derivatives: novel templates as potential antitumor agents.

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19 August 2018

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19 August 2018

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19 August 2018

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The Conformation ofcyclo(−d-Pro−Ala4−) as a Model for Cyclic Pentapeptides of thedL4Type

19 August 2018

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Pseudoprolines (Pro) in Drug Design: Direct Insertion of Pro Systems into Cyclosporin C

2 December 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/22287031

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.TET.2011.11.089

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21 January 2020

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21 January 2020

PubMed publication ID

22287031

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