Molecular mechanisms of Cys-loop ion channel receptor modulation by ivermectin. (Q35937704)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22586367%20AND%20SRC:MED&resulttype=core&format=json

1 February 2020

title

Molecular mechanisms of Cys-loop ion channel receptor modulation by ivermectin (English)

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1 February 2020

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1

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1 February 2020

author name string

Joseph W Lynch

series ordinal

2

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publication date

7 May 2012

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Frontiers in Molecular Neuroscience

1 February 2020

published in

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volume

5

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1 February 2020

page(s)

60

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Natural variation in a chloride channel subunit confers avermectin resistance in C. elegans

1 February 2020

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2 October 2017

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24 September 2018

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24 September 2018

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24 September 2018

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Mutations in the extracellular domains of glutamate-gated chloride channel alpha3 and beta subunits from ivermectin-resistant Cooperia oncophora affect agonist sensitivity

24 September 2018

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Selective elimination of glutamate activation and introduction of fluorescent proteins into a Caenorhabditis elegans chloride channel

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Identification of two novel Drosophila melanogaster histamine-gated chloride channel subunits expressed in the eye.

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24 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3345530

Activation of rat recombinant alpha(1)beta(2)gamma(2S) GABA(A) receptor by the insecticide ivermectin.

24 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3345530

Avermectin B1a binds to high- and low-affinity sites with dual effects on the gamma-aminobutyric acid-gated chloride channel of cultured cerebellar granule neurons.

24 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3345530

Environmental assessment of avermectins by the US Food and Drug Administration

24 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3345530

Ivermectin for spasticity in spinal-cord injury.

24 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3345530

Identification of acetylcholine receptor channel-lining residues in the entire M2 segment of the alpha subunit

24 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3345530

GABAA receptor needs two homologous domains of the beta-subunit for activation by GABA but not by pentobarbital

24 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3345530

Avermectin B1aModulation of ?-Aminobutyric Acid Receptors in Rat Brain Membranes

24 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3345530

Rings of negatively charged amino acids determine the acetylcholine receptor channel conductance

24 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3345530

Acetylcholine receptor channel imaged in the open state

24 September 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/22586367

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.3389/FNMOL.2012.00060

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22586367%20AND%20SRC:MED&resulttype=core&format=json

1 February 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22586367%20AND%20SRC:MED&resulttype=core&format=json

1 February 2020

PubMed publication ID

22586367

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22586367%20AND%20SRC:MED&resulttype=core&format=json